Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ RORγt Inverse Agonist II, GSK805
A cell-permeable, potent, non-toxic, inverse agonist of RORγt. Directly and reversibly interacts with the ligand binding domain of RORγt to block its transcriptional effects.
MilliporeSigma™ Calbiochem™ PP1 Analog II, 1NM-PP1
PP1 Analog II, CAS 221244-14-0, is a cell-permeable PP1 analog that acts as a potent, reversible, selective, ATP-competitive inhibitor of mutant over wild-type kinases.
MilliporeSigma™ Calbiochem™ Estrogen Receptor Antagonist, ICI 182,780
A cell-permeable estrogen antagonist. More effective than tamoxifen in reducing estrogen receptors in breast tumor cells.
MilliporeSigma™ Calbiochem™ AAA-ATPase Drg1 Inhibitor, Diazaborine
An anti-bacterial compound that targets NAD(P)H-dependent enoyl acyl carrier protein reductase (ENR) resulting in the inhibition of bacterial fatty acid synthase.
MilliporeSigma™ Calbiochem™ NMD Inhibitor
A cell-permeable inhibitor of nonsense-mediated mRNA decay (NMD) that enhances the stability of premature termination codon mutated p53 mRNA in N417 and HDQP-1 cells.
MilliporeSigma™ Calbiochem™ Piperlongumine
A cell-permeable, orally bioavailable natural product isolated from the plant species, Piper longum L, which selectively induces cell death in cancer cells that express both wild-type and mutant p53.
MilliporeSigma™ Calbiochem™ Proteasome Inhibitor Set I
The Proteasome Inhibitor Set I controls the biological activity of Proteasome. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ Protease Inhibitor Set
The Protease Inhibitor Set controls the activity of Protease. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ RAGE Antagonist Peptide, RAP
The RAGE Antagonist Peptide, RAP controls the biological activity of RAGE.
MilliporeSigma™ Calbiochem™ PTP1B Inhibitor
PTP1B Inhibitor, CAS 765317-72-4, is a cell-permeable, selective, reversible and non-competitive allosteric inhibitor of PTP1B (IC50 = 4 μM and 8 μM for PTP1B403 and PTP1B298, respectively).
MilliporeSigma™ Calbiochem™ PTP Inhibitor IV
The PTP Inhibitor IV, also referenced under CAS 329317-98-8, controls the biological activity of PTP. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
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MilliporeSigma™ Calbiochem™ Proteasome Substrate II, Fluorogenic
Fluorogenic proteasome substrate.
MilliporeSigma™ Calbiochem™ Protease Inhibitor Cocktail Set VII
Protease Inhibitor Cocktail Set VII contains five protease inhibitors with broad specificity. Recommended for purification of proteins containing His·Tag™ sequences.
MilliporeSigma™ Calbiochem™ Quinacrine, Dihydrochloride
A non-specific phospholipase A2 (PLA2) inhibitor.
MilliporeSigma™ Calbiochem™ Quercetin, Dihydrate
A cell-permeable and reversible inhibitor of PIM1 kinase (IC50 = 43nM), PI 3-K (IC50 = 3.8μM) and phospholipase A2